Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
5899 | 2283 | None | 0 | Rat | Binding | pKd | = | 8.8 | 8.8 | - | 1 | Guide to Pharmacology | None | None | None | None | 21724987 | |||||
5898 | 2374 | None | 0 | Rat | Binding | pKd | = | 9.6 | 9.6 | - | 1 | Guide to Pharmacology | None | None | None | None | 12782639 | |||||
5897 | 362 | None | 0 | Rat | Binding | pKd | = | 9.7 | 9.7 | 7 | 2 | Guide to Pharmacology | None | None | None | None | 12782639 | |||||
5897 | 362 | None | 0 | Rat | Binding | pKd | = | 9.7 | 9.7 | 7 | 2 | Guide to Pharmacology | None | None | None | None | 9208860 |